MUMBAI, India, June 26 -- Intellectual Property India has published a patent application (202443100315 A) filed by Neuland Laboratories Limited on December 18, 2024, for An Improved Process For The Preparation Of Tirzepatide Linker.
Inventors include Dr. Sharadsrikar Venkatesan Kotturi; Dr. Gandavadi Sunil Kumar; Mr. Parumanchala Shaik Shavali; Mr. Telakala Hema Sundara Rao; Mr. Shaik Kalesha; and Mr. Ramesh Reddy Filed On.
The application for the patent was published on June 19, 2026, under issue no. 25/2026.
Abstract: An improved process for the preparation of Tirzepatide having the chemical structural Formula I. The present invention also relates to the compounds of SEQ ID NO. 1 to 14 or a pharmaceutically acceptable salt thereof for use in the synthesis of Tirzepatide or a pharmaceutically acceptable salt thereof. The present invention further relates to the intermediate compounds of Formulae II to Formulae XVIII and their preparation process, which are used in the preparation of Tirzepatide or a pharmaceutically acceptable salt thereof. The present invention further relates to the process for preparing the Tirzepatide linker (SEQ ID NO. 3), its intermediate compounds of Formulae A to Formulae D and their preparation process, which are used in the preparation of the Tirzepatide linker (SEQ ID NO. 3).
Disclaimer: Curated by HT Syndication.